农药学学报2012，Vol.14Issue(6)：602-606,5.DOI:10.3969/j.issn.1008-7303.2012.06.03
N-[4-叔丁基-6-芳基-5-(1,2,4-三唑-1-基)-1,3-噻嗪-2-基]酰胺类化合物的合成及抑菌活性
Synthesis and antifungal activity of novel N-[4-tert-butyl-6-aryl-5-(1,2,4-triazol-1-yl)-1,3-thiazin-2-yl] amides
胡雷 1张妍妍 1席拓 1张毅文 1周文明1
作者信息
- 1. 西北农林科技大学理学院,陕西杨凌712100
- 折叠
摘要
Abstract
15 Novel compounds were synthesized from α-triazole pinacolone by condensation reaction, cyclization reaction and amidation reaction. Their structures were confirmed by IR,'H NMR and MS. The preliminary bioassay showed that all of the synthesized compounds have different inhibition on six tested plant pathogenic fungi at the concentration of 50 mg/L. The inhibition rates of compound 3a-3, 3a-4,3a-5,3b-2 and 3b-3 against Botrytis cinerea were up to 80%. 3a-4 and 3a-5 were 78. 6% and 82.4% against Fusarium oxysporum vasinfectum respectively.关键词
三唑/噻嗪/酰胺/合成/抑菌活性Key words
triazole/ thiazine/ amide/ synthesis/fungicidal activity分类
化学化工引用本文复制引用
胡雷,张妍妍,席拓,张毅文,周文明..N-[4-叔丁基-6-芳基-5-(1,2,4-三唑-1-基)-1,3-噻嗪-2-基]酰胺类化合物的合成及抑菌活性[J].农药学学报,2012,14(6):602-606,5.
