摘要
Abstract
As a bioisostere of diazoxide-based pharmaceuticals,benzo[e][1,2,3]oxathiazine-2,2-dioxides enable significant ability to improve pharmacokinetic properties of corresponding drugs and exhibit diverse biological activities,including antiviral,anticancer,anticonvulsant,and anti-osteoporosis effects.Consequently,research on their derivatization reactions has been increasing.This article focuses on the C-H bond functionalization of benzo[e][1,2,3]oxathiazine-2,2-dioxides and summarizes its reaction types as well as corresponding mechanisms.关键词
苯并[e][1,2,3]噁噻嗪-2,2-二氧化物/生物电子等排体/碳氢键官能团化Key words
benzo[e][1,2,3]oxathiazine-2,2-dioxide/bioisostere/C-H bond functionalization
